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HA-1077

●Purchase●DescriptionDihydrochlorideformofHA-1077

  • 产品型号:27030
  • 厂商性质:生产厂家
  • 更新时间:2024-01-31
  • 访  问  量:96
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Description

Dihydrochloride form of HA-1077. Inhibits a number of kinases, including ROCK I (IC50 = 10.7 µM), ROCK II (IC50 = 1.9 µM), MAPK1 (IC50 = 5 µM), and PKCRK2 (IC50 = 4 µM). Weaker inhibitor of PKC (IC50 = 425 µM) and MLCK (IC50 = 95 µM) .

This product has been cited 2 times.

Synonyms
Fasudil, Dihydrochloride Salt, 1-(5-Isoquinolinesulfonyl)homopiperazine, 2HCl, Eril, AT-877
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