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CHIR-99021 (CT99021) HCl

●Purchase●DescriptionCHIR-99021isahighlyspecificglycogensynthasekinase-3(GSK-3)inhibitorwhichcaninhibitbothisoformswithIC50of10nM(GSK-3α)and6

  • 产品型号:27615-3
  • 厂商性质:生产厂家
  • 更新时间:2024-01-31
  • 访  问  量:141
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Description

CHIR-99021 is a highly specific glycogen synthase kinase-3 (GSK-3) inhibitor which can inhibit both isoforms with IC50 of 10 nM (GSK-3α) and 6.7 nM (GSK-3β).

Synonyms
CHIR-99021; CT99021; 6-((2-((4-(2,4-dichlorophenyl)-5-(5-methyl-1H-imidazol-2-yl)pyrimidin-2-yl)amino)ethyl)amino)nicotinonitrile hydrochloride
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